Short Course



6:30 Dinner Workshop: Emerging Methods for Measuring Target Engagement*

The increase in usage of small molecule probes for the validation of novel therapeutic targets requires effective means of assaying target engagement in living systems. Importantly, measuring the extent to which a target is engaged (or not) provides critical information regarding probe selectivity and attributed efficacy modulating a biological process, while informing of any off-target interactions and potential toxicity. The workshop is designed to discuss emerging techniques and technologies for measuring target engagement.

Instructors: 

 

Erik Hett, Ph.D., Senior Scientist, Chemical Biology, Medicinal Chemistry, Pfizer

 

Thomas Lundbäck, Ph.D., Assay Development & Screening, Chemical Biology Consortium Sweden; Senior Scientist, Division of Translational Medicine & Chemical Biology, Department of Medical Biochemistry & Biophysics, Karolinska Institutet

 

Michael Dabrowski, Ph.D., CEO & Co-Founder, Pelago Bioscience AB

 

Andrea M. Zuhl, Ph.D., Fellow, Neuroscience, Pfizer; Former Research Associate, Cravatt Lab, The Scripps Research Institute

 

 


*Separate Registration Required


Download Brochure

2014 Chemical Biology for Target Validation Brochure 

Co-located Event

Structure Based Drug Design Co-Located 

Property Based Drug Design Colocaated Event 

Mastering Medicinal Chemistry 

WPC Colocated Event  

 


By Series:
By Region:


Conference
& Course Catalog

CHI Catalog 


Short Course DVDs